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| Title | Structure-Activity Relationships and Antileukemia Effects of the Tricyclic Benzoic Acid FTO Inhibitors. |
|---|---|
| Journal, issue, pages | J. Med. Chem., Vol. 65, Page 10638-10654, Year 2022 |
| Publish date | Dec 20, 2021 (structure data deposition date) |
Authors | Liu, Z. / Duan, Z. / Zhang, D. / Xiao, P. / Zhang, T. / Xu, H. / Wang, C.H. / Rao, G.W. / Gan, J. / Huang, Y. ...Liu, Z. / Duan, Z. / Zhang, D. / Xiao, P. / Zhang, T. / Xu, H. / Wang, C.H. / Rao, G.W. / Gan, J. / Huang, Y. / Yang, C.G. / Dong, Z. |
External links | J. Med. Chem. / PubMed:35793358 |
| Methods | X-ray diffraction |
| Resolution | 2.3 Å |
| Structure data | ![]() PDB-7wcv: |
| Chemicals | ![]() ChemComp-AKG: ![]() ChemComp-MN: ![]() ChemComp-943: ![]() ChemComp-HOH: |
| Source |
|
Keywords | OXIDOREDUCTASE / RNA demethylase / RNA BINDING PROTEIN |
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