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Title | Reversible lysine-targeted probes reveal residence time-based kinase selectivity. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 18, Page 934-941, Year 2022 |
Publish date | Jul 31, 2021 (structure data deposition date) |
Authors | Yang, T. / Cuesta, A. / Wan, X. / Craven, G.B. / Hirakawa, B. / Khamphavong, P. / May, J.R. / Kath, J.C. / Lapek Jr., J.D. / Niessen, S. ...Yang, T. / Cuesta, A. / Wan, X. / Craven, G.B. / Hirakawa, B. / Khamphavong, P. / May, J.R. / Kath, J.C. / Lapek Jr., J.D. / Niessen, S. / Burlingame, A.L. / Carelli, J.D. / Taunton, J. |
External links | Nat. Chem. Biol. / PubMed:35590003 |
Methods | X-ray diffraction |
Resolution | 2.32 Å |
Structure data | PDB-7fic: |
Chemicals | ChemComp-5YZ: ChemComp-CL: ChemComp-HOH: |
Source |
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Keywords | CELL CYCLE / Reversible lysine-targeted inhibitors; kinase |