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-Structure paper
Title | Discovery of a Novel Class of d-Amino Acid Oxidase Inhibitors Using the Schrodinger Computational Platform. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 6775-6802, Year 2022 |
Publish date | Mar 11, 2022 (structure data deposition date) |
![]() | Tang, H. / Jensen, K. / Houang, E. / McRobb, F.M. / Bhat, S. / Svensson, M. / Bochevarov, A. / Day, T. / Dahlgren, M.K. / Bell, J.A. ...Tang, H. / Jensen, K. / Houang, E. / McRobb, F.M. / Bhat, S. / Svensson, M. / Bochevarov, A. / Day, T. / Dahlgren, M.K. / Bell, J.A. / Frye, L. / Skene, R.J. / Lewis, J.H. / Osborne, J.D. / Tierney, J.P. / Gordon, J.A. / Palomero, M.A. / Gallati, C. / Chapman, R.S.L. / Jones, D.R. / Hirst, K.L. / Sephton, M. / Chauhan, A. / Sharpe, A. / Tardia, P. / Dechaux, E.A. / Taylor, A. / Waddell, R.D. / Valentine, A. / Janssens, H.B. / Aziz, O. / Bloomfield, D.E. / Ladha, S. / Fraser, I.J. / Ellard, J.M. |
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Methods | X-ray diffraction |
Resolution | 1.66 - 2.1 Å |
Structure data | ![]() PDB-7u9s: ![]() PDB-7u9u: |
Chemicals | ![]() ChemComp-FAD: ![]() ChemComp-M7I: ![]() ChemComp-HOH: ![]() ChemComp-BEZ: ![]() ChemComp-M89: |
Source |
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![]() | OXIDOREDUCTASE/INHIBITOR / FAD / Flavoprotein / Oxidoreductase / Peroxisome / OXIDOREDUCTASE-INHIBITOR complex |