タイトル | Structural basis for replicase polyprotein cleavage and substrate specificity of main protease from SARS-CoV-2. |
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ジャーナル・号・ページ | Proc. Natl. Acad. Sci. USA, Vol. 119, Page e2117142119-e2117142119, Year 2022 |
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掲載日 | 2020年2月19日 (構造データの登録日) |
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著者 | Zhao, Y. / Zhu, Y. / Liu, X. / Jin, Z. / Duan, Y. / Zhang, Q. / Wu, C. / Feng, L. / Du, X. / Zhao, J. ...Zhao, Y. / Zhu, Y. / Liu, X. / Jin, Z. / Duan, Y. / Zhang, Q. / Wu, C. / Feng, L. / Du, X. / Zhao, J. / Shao, M. / Zhang, B. / Yang, X. / Wu, L. / Ji, X. / Guddat, L.W. / Yang, K. / Rao, Z. / Yang, H. |
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リンク | Proc. Natl. Acad. Sci. USA / PubMed:35380892 |
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手法 | X線回折 |
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解像度 | 1.49 - 2.19 Å |
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構造データ | PDB-6m03: The crystal structure of COVID-19 main protease in apo form 手法: X-RAY DIFFRACTION / 解像度: 2.0 Å PDB-7dvp: SARS-CoV-2 Mpro mutant (H41A) in complex with nsp4|5 peptidyl substrate 手法: X-RAY DIFFRACTION / 解像度: 1.69 Å PDB-7dvw: SARS-CoV-2 Mpro mutant (H41A) in complex with nsp5|6 peptidyl substrate 手法: X-RAY DIFFRACTION / 解像度: 1.49 Å PDB-7dvx: SARS-CoV-2 Mpro mutant (H41A) in complex with nsp6|7 peptidyl substrate 手法: X-RAY DIFFRACTION / 解像度: 1.8 Å PDB-7dvy: SARS-CoV-2 Mpro mutant (H41A) in complex with nsp9|10 peptidyl substrate 手法: X-RAY DIFFRACTION / 解像度: 1.8 Å PDB-7dw0: SARS-CoV-2 Mpro mutant (H41A) in complex with nsp14|15 peptidyl substrate 手法: X-RAY DIFFRACTION / 解像度: 1.81 Å PDB-7dw6: SARS-CoV-2 Mpro mutant (H41A) in complex with nsp15|16 peptidyl substrate 手法: X-RAY DIFFRACTION / 解像度: 1.7 Å PDB-7e5x: THE CRYSTAL STRUCTURE OF COVID-19 MAIN PROTEASE apo form at 2.2 angstrom 手法: X-RAY DIFFRACTION / 解像度: 2.19 Å PDB-7vah: The crystal structure of COVID-19 main protease in H41A mutation 手法: X-RAY DIFFRACTION / 解像度: 1.491 Å |
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化合物 | |
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由来 | ![](img/tx_virus.gif) severe acute respiratory syndrome coronavirus 2 (ウイルス)
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キーワード | BIOSYNTHETIC PROTEIN / Coronavirus / COVID-19 / viral protease / VIRAL PROTEIN / protease |
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