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-Structure paper
Title | Discovery of a highly potent CECR2 bromodomain inhibitor with 7H-pyrrolo[2,3-d] pyrimidine scaffold. |
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Journal, issue, pages | Bioorg. Chem., Vol. 123, Page 105768-105768, Year 2022 |
Publish date | Sep 6, 2021 (structure data deposition date) |
![]() | Lu, H. / Lu, T. / Zu, S. / Duan, Z. / Guang, Y. / Li, Q. / Ma, J. / Chen, D. / Li, B. / Lu, W. ...Lu, H. / Lu, T. / Zu, S. / Duan, Z. / Guang, Y. / Li, Q. / Ma, J. / Chen, D. / Li, B. / Lu, W. / Jiang, H. / Luo, C. / Ye, D. / Chen, K. / Lin, H. |
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Methods | X-ray diffraction |
Resolution | 1.85659146555 Å |
Structure data | ![]() PDB-7vd4: |
Chemicals | ![]() ChemComp-6FI: ![]() ChemComp-HOH: |
Source |
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![]() | ANTITUMOR PROTEIN / BPTF Bromodomain / Lysine acetylation / small-molecule inhibitor / BIOSYNTHETIC PROTEIN |