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-Structure paper
Title | Optimization of Brigatinib as New Wild-Type Sparing Inhibitors of EGFR T790M/C797S Mutants. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 13, Page 196-202, Year 2022 |
Publish date | May 5, 2021 (structure data deposition date) |
![]() | Li, S. / Zhang, T. / Zhu, S.J. / Lei, C. / Lai, M. / Peng, L. / Tong, L. / Pang, Z. / Lu, X. / Ding, J. ...Li, S. / Zhang, T. / Zhu, S.J. / Lei, C. / Lai, M. / Peng, L. / Tong, L. / Pang, Z. / Lu, X. / Ding, J. / Ren, X. / Yun, C.H. / Xie, H. / Ding, K. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.662 Å |
Structure data | ![]() PDB-7er2: |
Chemicals | ![]() ChemComp-JAU: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / EGFR / T790M/C797S / inhibitor |