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| Title | A Novel HER2-Selective Kinase Inhibitor Is Effective in HER2 Mutant and Amplified Non-Small Cell Lung Cancer. |
|---|---|
| Journal, issue, pages | Cancer Res., Vol. 82, Page 1633-1645, Year 2022 |
| Publish date | Aug 27, 2020 (structure data deposition date) |
Authors | Son, J. / Jang, J. / Beyett, T.S. / Eum, Y. / Haikala, H.M. / Verano, A. / Lin, M. / Hatcher, J.M. / Kwiatkowski, N.P. / Eser, P.O. ...Son, J. / Jang, J. / Beyett, T.S. / Eum, Y. / Haikala, H.M. / Verano, A. / Lin, M. / Hatcher, J.M. / Kwiatkowski, N.P. / Eser, P.O. / Poitras, M.J. / Wang, S. / Xu, M. / Gokhale, P.C. / Cameron, M.D. / Eck, M.J. / Gray, N.S. / Janne, P.A. |
External links | Cancer Res. / PubMed:35149586 |
| Methods | X-ray diffraction |
| Resolution | 3.27 Å |
| Structure data | ![]() PDB-7jxh: |
| Chemicals | ![]() ChemComp-VOY: |
| Source |
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Keywords | TRANSFERASE/TRANSFERASE Inhibitor / HER2 / ErbB2 / kinase / inhibitor / TRANSFERASE / TRANSFERASE-TRANSFERASE Inhibitor complex |
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homo sapiens (human)
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