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-Structure paper
Title | Discovery of Dimeric Arylsulfonamides as Potent ADAM8 Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 1787-1793, Year 2021 |
Publish date | Jun 15, 2021 (structure data deposition date) |
![]() | Cuffaro, D. / Camodeca, C. / Tuccinardi, T. / Ciccone, L. / Bartsch, J.W. / Kellermann, T. / Cook, L. / Nuti, E. / Rossello, A. |
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Methods | X-ray diffraction |
Resolution | 1.24 Å |
Structure data | ![]() PDB-7ovy: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-CA: ![]() ChemComp-2IF: ![]() ChemComp-EDO: ![]() ChemComp-PGR: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/HYDROLASE INHIBITOR / Hydrolase / Hydrolase-Inhibitor crystal complex / HYDROLASE INHIBITOR / HYDROLASE-HYDROLASE INHIBITOR complex |