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-Structure paper
Title | Novel Macrocyclic Peptidomimetics Targeting the Polo-Box Domain of Polo-Like Kinase 1. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 1915-1932, Year 2022 |
Publish date | May 11, 2021 (structure data deposition date) |
Authors | Ryu, S. / Park, J.E. / Ham, Y.J. / Lim, D.C. / Kwiatkowski, N.P. / Kim, D.H. / Bhunia, D. / Kim, N.D. / Yaffe, M.B. / Son, W. ...Ryu, S. / Park, J.E. / Ham, Y.J. / Lim, D.C. / Kwiatkowski, N.P. / Kim, D.H. / Bhunia, D. / Kim, N.D. / Yaffe, M.B. / Son, W. / Kim, N. / Choi, T.I. / Swain, P. / Kim, C.H. / Lee, J.Y. / Gray, N.S. / Lee, K.S. / Sim, T. |
External links | J. Med. Chem. / PubMed:35029981 |
Methods | X-ray diffraction |
Resolution | 1.85 Å |
Structure data | PDB-7mso: |
Chemicals | ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/Inhibitor / phosphopeptide binding domain / TRANSFERASE-Inhibitor complex |