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-Structure paper
Title | Dihydropyridine Lactam Analogs Targeting BET Bromodomains. |
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Journal, issue, pages | Chemmedchem, Vol. 17, Page e202100407-e202100407, Year 2022 |
Publish date | Jan 21, 2021 (structure data deposition date) |
Authors | Jiang, J. / Sigua, L.H. / Chan, A. / Kalra, P. / Pomerantz, W.C.K. / Schonbrunn, E. / Qi, J. / Georg, G.I. |
External links | Chemmedchem / PubMed:34932262 |
Methods | X-ray diffraction |
Resolution | 1.75 Å |
Structure data | PDB-7lh8: |
Chemicals | ChemComp-XZG: ChemComp-EDO: ChemComp-NA: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION/INHIBITOR / Small molecule inhibitor / drug discovery / epigenetics / TRANSCRIPTION / TRANSCRIPTION-INHIBITOR complex |