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-Structure paper
Title | Potent and Selective RIPK1 Inhibitors Targeting Dual-Pockets for the Treatment of Systemic Inflammatory Response Syndrome and Sepsis. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 61, Page e202114922-e202114922, Year 2022 |
Publish date | Jul 15, 2021 (structure data deposition date) |
Authors | Yang, X. / Lu, H. / Xie, H. / Zhang, B. / Nie, T. / Fan, C. / Yang, T. / Xu, Y. / Su, H. / Tang, W. / Zhou, B. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:34851543 |
Methods | X-ray diffraction |
Resolution | 2 - 2.21 Å |
Structure data | PDB-7fcz: PDB-7fd0: |
Chemicals | ChemComp-3IF: ChemComp-HOH: ChemComp-3IU: |
Source |
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Keywords | IMMUNE SYSTEM/INHIBITOR / IMMUNE SYSTEM-INHIBITOR COMPLEX |