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-Structure paper
Title | Inhibitors of the Hippo Pathway Kinases STK3/MST2 and STK4/MST1 Have Utility for the Treatment of Acute Myeloid Leukemia. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 1352-1369, Year 2022 |
Publish date | Mar 13, 2020 (structure data deposition date) |
![]() | Bata, N. / Chaikuad, A. / Bakas, N.A. / Limpert, A.S. / Lambert, L.J. / Sheffler, D.J. / Berger, L.M. / Liu, G. / Yuan, C. / Wang, L. ...Bata, N. / Chaikuad, A. / Bakas, N.A. / Limpert, A.S. / Lambert, L.J. / Sheffler, D.J. / Berger, L.M. / Liu, G. / Yuan, C. / Wang, L. / Peng, Y. / Dong, J. / Celeridad, M. / Layng, F. / Knapp, S. / Cosford, N.D.P. |
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Methods | X-ray diffraction |
Resolution | 2.58 Å |
Structure data | ![]() PDB-6yat: |
Chemicals | ![]() ChemComp-3FX: ![]() ChemComp-GOL: ![]() ChemComp-OJ5: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE / kinase / kinase inhibitor / MST1 / STK4 / hippo pathway / chemical probe / Structural Genomics / Structural Genomics Consortium / SGC |