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-Structure paper
Title | From Fragment to Lead: De Novo Design and Development toward a Selective FGFR2 Inhibitor. |
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Journal, issue, pages | J. Med. Chem., Vol. 65, Page 1481-1504, Year 2022 |
Publish date | Jun 27, 2021 (structure data deposition date) |
Authors | Turner, L.D. / Trinh, C.H. / Hubball, R.A. / Orritt, K.M. / Lin, C.C. / Burns, J.E. / Knowles, M.A. / Fishwick, C.W.G. |
External links | J. Med. Chem. / PubMed:34780700 |
Methods | X-ray diffraction |
Resolution | 1.71 - 2.28 Å |
Structure data | PDB-7ozb: PDB-7ozd: PDB-7ozf: PDB-7ozy: |
Chemicals | ChemComp-47I: ChemComp-SO4: ChemComp-EDO: ChemComp-HOH: ChemComp-42I: ChemComp-466: ChemComp-CL: |
Source |
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Keywords | TRANSFERASE / FGFR1 / Inhibitor / receptor tyrosine kinase / FGFR2 |