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-Structure paper
Title | An Ultrapotent and Selective Cyclic Peptide Inhibitor of Human beta-Factor XIIa in a Cyclotide Scaffold. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 143, Page 18481-18489, Year 2021 |
Publish date | Jul 12, 2021 (structure data deposition date) |
Authors | Liu, W. / de Veer, S.J. / Huang, Y.H. / Sengoku, T. / Okada, C. / Ogata, K. / Zdenek, C.N. / Fry, B.G. / Swedberg, J.E. / Passioura, T. ...Liu, W. / de Veer, S.J. / Huang, Y.H. / Sengoku, T. / Okada, C. / Ogata, K. / Zdenek, C.N. / Fry, B.G. / Swedberg, J.E. / Passioura, T. / Craik, D.J. / Suga, H. |
External links | J. Am. Chem. Soc. / PubMed:34723512 |
Methods | X-ray diffraction |
Resolution | 1.99 Å |
Structure data | PDB-7fbp: |
Chemicals | ChemComp-HOH: |
Source |
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Keywords | BLOOD CLOTTING / Serine protease / Inhibitor / macrocyclic peptide / Cyclotide |