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-Structure paper
Title | Development of BET inhibitors as potential treatments for cancer: A new carboline chemotype. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 51, Page 128376-128376, Year 2021 |
Publish date | Apr 2, 2021 (structure data deposition date) |
Authors | Hill, M.D. / Quesnelle, C. / Tokarski, J. / Fang, H. / Fanslau, C. / Haarhoff, Z. / Kramer, M. / Madari, S. / Wiebesiek, A. / Morrison, J. ...Hill, M.D. / Quesnelle, C. / Tokarski, J. / Fang, H. / Fanslau, C. / Haarhoff, Z. / Kramer, M. / Madari, S. / Wiebesiek, A. / Morrison, J. / Simmermacher-Mayer, J. / Sinz, M. / Westhouse, R. / Xie, C. / Zhao, J. / Huang, L. / Sheriff, S. / Yan, C. / Marsilio, F. / Everlof, G. / Zvyaga, T. / Lee, F. / Gavai, A.V. / Degnan, A.P. |
External links | Bioorg. Med. Chem. Lett. / PubMed:34560263 |
Methods | X-ray diffraction |
Resolution | 1.76 Å |
Structure data | PDB-7mce: |
Chemicals | ChemComp-YWY: ChemComp-HOH: |
Source |
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Keywords | CELL CYCLE / BROMODOMAIN-CONTAINING PROTEIN 4 ISOFORM LONG / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / CAP / HUNK1 / MCAP / MITOTIC CHROMOSOME ASSOCIATED PROTEIN SGC |