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-Structure paper
Title | Pan-3C Protease Inhibitor Rupintrivir Binds SARS-CoV-2 Main Protease in a Unique Binding Mode. |
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Journal, issue, pages | Biochemistry, Vol. 60, Page 2925-2931, Year 2021 |
Publish date | Dec 31, 2020 (structure data deposition date) |
![]() | Lockbaum, G.J. / Henes, M. / Lee, J.M. / Timm, J. / Nalivaika, E.A. / Thompson, P.R. / Kurt Yilmaz, N. / Schiffer, C.A. |
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Methods | X-ray diffraction |
Resolution | 1.95 - 2.45 Å |
Structure data | ![]() PDB-7l8h: ![]() PDB-7l8i: ![]() PDB-7l8j: |
Chemicals | ![]() ChemComp-AG7: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/INHIBITOR / ENTEROVIRUS / EV68 / PROTEASE / PROTEASE INHIBITOR / COMPLEX / HYDROLASE INHIBITOR COMPLEX / HYDROLASE / HYDROLASE-HYDROLASE INHIBITOR COMPLEX / RUPINTRIVIR / HYDROLASE-INHIBITOR complex / SARS-CoV-2 / SARS2 / COVID19 |