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-Structure paper
Title | DNA-encoded chemistry technology yields expedient access to SARS-CoV-2 M pro inhibitors. |
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Journal, issue, pages | Proc. Natl. Acad. Sci. USA, Vol. 118, Year 2021 |
Publish date | Feb 19, 2021 (structure data deposition date) |
![]() | Chamakuri, S. / Lu, S. / Ucisik, M.N. / Bohren, K.M. / Chen, Y.C. / Du, H.C. / Faver, J.C. / Jimmidi, R. / Li, F. / Li, J.Y. ...Chamakuri, S. / Lu, S. / Ucisik, M.N. / Bohren, K.M. / Chen, Y.C. / Du, H.C. / Faver, J.C. / Jimmidi, R. / Li, F. / Li, J.Y. / Nyshadham, P. / Palmer, S.S. / Pollet, J. / Qin, X. / Ronca, S.E. / Sankaran, B. / Sharma, K.L. / Tan, Z. / Versteeg, L. / Yu, Z. / Matzuk, M.M. / Palzkill, T. / Young, D.W. |
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Methods | X-ray diffraction |
Resolution | 1.79 Å |
Structure data | ![]() PDB-7ltn: |
Chemicals | ![]() ChemComp-YCV: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE/INHIBITOR / Sars-Cov-2 main protease / nanomolar potency inhibitor / DNA-encoded library / HYDROLASE-INHIBITOR complex |