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-Structure paper
Title | Discovery of a Novel Bromodomain and Extra Terminal Domain (BET) Protein Inhibitor, I-BET282E, Suitable for Clinical Progression. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 12200-12227, Year 2021 |
Publish date | Mar 28, 2021 (structure data deposition date) |
![]() | Jones, K.L. / Beaumont, D.M. / Bernard, S.G. / Bit, R.A. / Campbell, S.P. / Chung, C.W. / Cutler, L. / Demont, E.H. / Dennis, K. / Gordon, L. ...Jones, K.L. / Beaumont, D.M. / Bernard, S.G. / Bit, R.A. / Campbell, S.P. / Chung, C.W. / Cutler, L. / Demont, E.H. / Dennis, K. / Gordon, L. / Gray, J.R. / Haase, M.V. / Lewis, A.J. / McCleary, S. / Mitchell, D.J. / Moore, S.M. / Parr, N. / Robb, O.J. / Smithers, N. / Soden, P.E. / Suckling, C.J. / Taylor, S. / Walker, A.L. / Watson, R.J. / Prinjha, R.K. |
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Methods | X-ray diffraction |
Resolution | 1.7 Å |
Structure data | ![]() PDB-7o18: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-UYK: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / INHIBITOR / HISTONE / EPIGENETIC READER / BROMODOMAIN / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / ANTAGONIST |