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-Structure paper
Title | Efficient Entropy-Driven Inhibition of Dipeptidyl Peptidase III by Hydroxyethylene Transition-State Peptidomimetics. |
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Journal, issue, pages | Chemistry, Vol. 27, Page 14108-14120, Year 2021 |
Publish date | Jun 12, 2021 (structure data deposition date) |
![]() | Ivkovic, J. / Jha, S. / Lembacher-Fadum, C. / Puschnig, J. / Kumar, P. / Reithofer, V. / Gruber, K. / Macheroux, P. / Breinbauer, R. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.65 Å |
Structure data | ![]() PDB-7oup: |
Chemicals | ![]() ChemComp-ZN: ![]() ChemComp-K: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
Source |
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![]() | HYDROLASE / Inhibitor / COMPLEX / PEPTIDASE / ZINC-HYDROLASE |