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-Structure paper
Title | M3258 Is a Selective Inhibitor of the Immunoproteasome Subunit LMP7 ( beta 5i) Delivering Efficacy in Multiple Myeloma Models. |
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Journal, issue, pages | Mol. Cancer Ther., Vol. 20, Page 1378-1387, Year 2021 |
Publish date | Nov 6, 2020 (structure data deposition date) |
![]() | Sanderson, M.P. / Friese-Hamim, M. / Walter-Bausch, G. / Busch, M. / Gaus, S. / Musil, D. / Rohdich, F. / Zanelli, U. / Downey-Kopyscinski, S.L. / Mitsiades, C.S. ...Sanderson, M.P. / Friese-Hamim, M. / Walter-Bausch, G. / Busch, M. / Gaus, S. / Musil, D. / Rohdich, F. / Zanelli, U. / Downey-Kopyscinski, S.L. / Mitsiades, C.S. / Schadt, O. / Klein, M. / Esdar, C. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.288 Å |
Structure data | ![]() PDB-7awe: |
Chemicals | ![]() ChemComp-NA: ![]() ChemComp-SCN: ![]() ChemComp-S5K: ![]() ChemComp-HOH: |
Source |
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![]() | IMMUNE SYSTEM / MULTICATALYTIC PROTEINASE / 20S PROTEASOME / PROTEASE / HYDROLASE |