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-Structure paper
Title | Development of BET inhibitors as potential treatments for cancer: A search for structural diversity. |
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Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 44, Page 128108-128108, Year 2021 |
Publish date | Apr 2, 2021 (structure data deposition date) |
Authors | Hill, M.D. / Fang, H. / Tokarski, J. / Fanslau, C. / Haarhoff, Z. / Huang, C. / Kramer, M. / Menard, K. / Monereau, L. / Morrison, J. ...Hill, M.D. / Fang, H. / Tokarski, J. / Fanslau, C. / Haarhoff, Z. / Huang, C. / Kramer, M. / Menard, K. / Monereau, L. / Morrison, J. / Ranasinghe, A. / Shields, E.E. / Tye, C.K. / Westhouse, R. / Everlof, G. / Sheriff, S. / Yan, C. / Marsilio, F. / Zhang, L. / Zvyaga, T. / Lee, F. / Gavai, A.V. / Degnan, A.P. |
External links | Bioorg. Med. Chem. Lett. / PubMed:33991625 |
Methods | X-ray diffraction |
Resolution | 2.19 Å |
Structure data | PDB-7mcf: |
Chemicals | ChemComp-YX4: ChemComp-HOH: |
Source |
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Keywords | CELL CYCLE / BROMODOMAIN-CONTAINING PROTEIN 4 ISOFORM LONG / BRD4 / BROMODOMAIN CONTAINING PROTEIN 4 / CAP / HUNK1 / MCAP / MITOTIC CHROMOSOME ASSOCIATED PROTEIN SGC |