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Title | 7-(2-Anilinopyrimidin-4-yl)-1-benzazepin-2-ones Designed by a "Cut and Glue" Strategy Are Dual Aurora A/VEGF-R Kinase Inhibitors. |
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Journal, issue, pages | Molecules, Vol. 26, Year 2021 |
Publish date | Nov 12, 2020 (structure data deposition date) |
Authors | Karatas, M. / Chaikuad, A. / Berger, B. / Kubbutat, M.H.G. / Totzke, F. / Knapp, S. / Kunick, C. |
External links | Molecules / PubMed:33799460 |
Methods | X-ray diffraction |
Resolution | 2.8 - 2.86 Å |
Structure data | PDB-7ayh: PDB-7ayi: |
Chemicals | ChemComp-S9H: ChemComp-S9K: |
Source |
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Keywords | TRANSFERASE / kinase / kinase inhibitor / aurora kinase / stk6 / Structural Genomics / Structural Genomics Consortium / SGC |