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-Structure paper
Title | Structure-Enabled Discovery of Novel Macrocyclic Inhibitors Targeting Glutaminase 1 Allosteric Binding Site. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 4588-4611, Year 2021 |
Publish date | Jan 7, 2020 (structure data deposition date) |
Authors | Xu, X. / Wang, J. / Wang, M. / Yuan, X. / Li, L. / Zhang, C. / Huang, H. / Jing, T. / Wang, C. / Tong, C. ...Xu, X. / Wang, J. / Wang, M. / Yuan, X. / Li, L. / Zhang, C. / Huang, H. / Jing, T. / Wang, C. / Tong, C. / Zhou, L. / Meng, Y. / Xu, P. / Kou, J. / Qiu, Z. / Li, Z. / Bian, J. |
External links | J. Med. Chem. / PubMed:33792311 |
Methods | X-ray diffraction |
Resolution | 3.2 Å |
Structure data | PDB-6lox: |
Chemicals | ChemComp-EN3: ChemComp-HOH: |
Source |
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Keywords | PROTEIN BINDING / protein-inhibitor complex |