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-Structure paper
Title | Structure-Based Exploration of Selectivity for ATM Inhibitors in Huntington's Disease. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 5018-5036, Year 2021 |
Publish date | Apr 6, 2020 (structure data deposition date) |
Authors | Van de Poel, A. / Toledo-Sherman, L. / Breccia, P. / Cachope, R. / Bate, J.R. / Angulo-Herrera, I. / Wishart, G. / Matthews, K.L. / Martin, S.L. / Peacock, M. ...Van de Poel, A. / Toledo-Sherman, L. / Breccia, P. / Cachope, R. / Bate, J.R. / Angulo-Herrera, I. / Wishart, G. / Matthews, K.L. / Martin, S.L. / Peacock, M. / Barnard, A. / Cox, H.C. / Jones, G. / McAllister, G. / Vater, H. / Esmieu, W. / Clissold, C. / Lamers, M. / Leonard, P. / Jarvis, R.E. / Blackaby, W. / Eznarriaga, M. / Lazari, O. / Yates, D. / Rose, M. / Jang, S.W. / Munoz-Sanjuan, I. / Dominguez, C. |
External links | J. Med. Chem. / PubMed:33783225 |
Methods | X-ray diffraction |
Resolution | 3.12 Å |
Structure data | PDB-6ykg: |
Chemicals | ChemComp-OZ8: ChemComp-HOH: |
Source |
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Keywords | LYASE / Huntingtons disease; VPS34 / ATM |