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-Structure paper
Title | Virtual Screening Approach to Identifying a Novel and Tractable Series of Pseudomonas aeruginosa Elastase Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 217-227, Year 2021 |
Publish date | Sep 29, 2020 (structure data deposition date) |
Authors | Leiris, S. / Davies, D.T. / Sprynski, N. / Castandet, J. / Beyria, L. / Bodnarchuk, M.S. / Sutton, J.M. / Mullins, T.M.G. / Jones, M.W. / Forrest, A.K. ...Leiris, S. / Davies, D.T. / Sprynski, N. / Castandet, J. / Beyria, L. / Bodnarchuk, M.S. / Sutton, J.M. / Mullins, T.M.G. / Jones, M.W. / Forrest, A.K. / Pallin, T.D. / Karunakar, P. / Martha, S.K. / Parusharamulu, B. / Ramula, R. / Kotha, V. / Pottabathini, N. / Pothukanuri, S. / Lemonnier, M. / Everett, M. |
External links | Acs Med. Chem. Lett. / PubMed:33603968 |
Methods | X-ray diffraction |
Resolution | 1.75 Å |
Structure data | PDB-7ajr: |
Chemicals | ChemComp-RJB: ChemComp-ZN: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | HYDROLASE / Pseudomonas aeruginosa / elastase / inhibitors |