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-Structure paper
Title | A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 3697-3706, Year 2021 |
Publish date | Mar 16, 2020 (structure data deposition date) |
Authors | Shen, Y. / Li, F. / Szewczyk, M.M. / Halabelian, L. / Chau, I. / Eram, M.S. / Dela Sena, C. / Park, K.S. / Meng, F. / Chen, H. ...Shen, Y. / Li, F. / Szewczyk, M.M. / Halabelian, L. / Chau, I. / Eram, M.S. / Dela Sena, C. / Park, K.S. / Meng, F. / Chen, H. / Zeng, H. / Dong, A. / Wu, H. / Trush, V.V. / McLeod, D. / Zepeda-Velazquez, C.A. / Campbell, R.M. / Mader, M.M. / Watson, B.M. / Schapira, M. / Arrowsmith, C.H. / Al-Awar, R. / Barsyte-Lovejoy, D. / Kaniskan, H.U. / Brown, P.J. / Vedadi, M. / Jin, J. |
External links | J. Med. Chem. / PubMed:33591753 |
Methods | X-ray diffraction |
Resolution | 1.91 Å |
Structure data | PDB-6w6d: |
Chemicals | ChemComp-SAH: ChemComp-T9A: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE Inhibitor / PRMT6 and SGC6870 inhibitor / Structural Genomics / Structural Genomics Consortium / SGC / TRANSFERASE / TRANSFERASE-TRANSFERASE Inhibitor complex |