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Title | Kinetics-Driven Drug Design Strategy for Next-Generation Acetylcholinesterase Inhibitors to Clinical Candidate. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 1844-1855, Year 2021 |
Publish date | Oct 14, 2020 (structure data deposition date) |
![]() | Zhou, Y. / Fu, Y. / Yin, W. / Li, J. / Wang, W. / Bai, F. / Xu, S. / Gong, Q. / Peng, T. / Hong, Y. ...Zhou, Y. / Fu, Y. / Yin, W. / Li, J. / Wang, W. / Bai, F. / Xu, S. / Gong, Q. / Peng, T. / Hong, Y. / Zhang, D. / Liu, Q. / Xu, Y. / Xu, H.E. / Zhang, H. / Jiang, H. / Liu, H. |
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Methods | X-ray diffraction |
Resolution | 2.45 - 2.85 Å |
Structure data | ![]() PDB-7d9o: ![]() PDB-7d9p: ![]() PDB-7d9q: |
Chemicals | ![]() ChemComp-H0L: ![]() ChemComp-HOH: ![]() ChemComp-H0R: ![]() ChemComp-H1R: |
Source |
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![]() | HYDROLASE / AchE inhibitor / complex structure |