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-Structure paper
Title | Discovery of a Novel Series of Potent and Selective Alkynylthiazole-Derived PI3K gamma Inhibitors. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 12, Page 129-135, Year 2021 |
Publish date | Oct 27, 2020 (structure data deposition date) |
![]() | Bandarage, U.K. / Aronov, A.M. / Cao, J. / Come, J.H. / Cottrell, K.M. / Davies, R.J. / Giroux, S. / Jacobs, M. / Mahajan, S. / Messersmith, D. ...Bandarage, U.K. / Aronov, A.M. / Cao, J. / Come, J.H. / Cottrell, K.M. / Davies, R.J. / Giroux, S. / Jacobs, M. / Mahajan, S. / Messersmith, D. / Moody, C.S. / Swett, R. / Xu, J. |
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Methods | X-ray diffraction |
Resolution | 2.81 Å |
Structure data | ![]() PDB-7kke: |
Chemicals | ![]() ChemComp-WJV: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/Inhibitor / KINASE / INHIBITOR / TRANSFERASE-Inhibitor complex |