+Search query
-Structure paper
Title | Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine Methyltransferase. |
---|---|
Journal, issue, pages | Chembiochem, Vol. 22, Page 1597-1608, Year 2021 |
Publish date | Apr 27, 2020 (structure data deposition date) |
![]() | Talibov, V.O. / Fabini, E. / FitzGerald, E.A. / Tedesco, D. / Cederfeldt, D. / Talu, M.J. / Rachman, M.M. / Mihalic, F. / Manoni, E. / Naldi, M. ...Talibov, V.O. / Fabini, E. / FitzGerald, E.A. / Tedesco, D. / Cederfeldt, D. / Talu, M.J. / Rachman, M.M. / Mihalic, F. / Manoni, E. / Naldi, M. / Sanese, P. / Forte, G. / Lepore Signorile, M. / Barril, X. / Simone, C. / Bartolini, M. / Dobritzsch, D. / Del Rio, A. / Danielson, U.H. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.93 Å |
Structure data | ![]() PDB-6yuh: |
Chemicals | ![]() ChemComp-SAM: ![]() ChemComp-GOL: ![]() ChemComp-POW: ![]() ChemComp-ZN: ![]() ChemComp-HOH: |
Source |
|
![]() | ONCOPROTEIN / Methyltransferase / complex / inhibitor |