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-Structure paper
Title | Diflunisal Derivatives as Modulators of ACMS Decarboxylase Targeting the Tryptophan-Kynurenine Pathway. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 797-811, Year 2021 |
Publish date | Sep 7, 2020 (structure data deposition date) |
Authors | Yang, Y. / Borel, T. / de Azambuja, F. / Johnson, D. / Sorrentino, J.P. / Udokwu, C. / Davis, I. / Liu, A. / Altman, R.A. |
External links | J. Med. Chem. / PubMed:33369426 |
Methods | X-ray diffraction |
Resolution | 1.83 - 2.17 Å |
Structure data | PDB-7k12: PDB-7k13: |
Chemicals | ChemComp-ZN: ChemComp-1FL: ChemComp-CIT: ChemComp-HOH: ChemComp-VR7: |
Source |
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Keywords | LYASE / FDA-approved drugs / NAD+ / neuropsychiatric disorders / decarboxylase |