+Search query
-Structure paper
Title | Discovery of novel HIV-1 integrase-LEDGF/p75 allosteric inhibitors based on a pyridine scaffold forming an intramolecular hydrogen bond. |
---|---|
Journal, issue, pages | Bioorg. Med. Chem. Lett., Vol. 33, Page 127742-127742, Year 2020 |
Publish date | Oct 7, 2020 (structure data deposition date) |
![]() | Sugiyama, S. / Akiyama, T. / Taoda, Y. / Iwaki, T. / Matsuoka, E. / Akihisa, E. / Seki, T. / Yoshinaga, T. / Kawasuji, T. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 2.43 Å |
Structure data | ![]() PDB-7d83: |
Chemicals | ![]() ChemComp-SO4: ![]() ChemComp-GZ9: ![]() ChemComp-HOH: |
Source |
|
![]() | VIRAL PROTEIN / HIV-1 Integrase |