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-Structure paper
Title | Development of a Potent and Specific FGFR4 Inhibitor for the Treatment of Hepatocellular Carcinoma. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 11484-11497, Year 2020 |
Publish date | Mar 26, 2019 (structure data deposition date) |
Authors | Rezende Miranda, R. / Fu, Y. / Chen, X. / Perino, J. / Cao, P. / Carpten, J. / Chen, Y. / Zhang, C. |
External links | J. Med. Chem. / PubMed:33030342 |
Methods | X-ray diffraction |
Resolution | 1.601 Å |
Structure data | PDB-6jpe: |
Chemicals | ChemComp-BYU: ChemComp-SO4: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE INHIBITOR / FGFR4 / irreversible inhibitor / TRANSFERASE-TRANSFERASE INHIBITOR complex |