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-Structure paper
Title | Selective N-Terminal BET Bromodomain Inhibitors by Targeting Non-Conserved Residues and Structured Water Displacement*. |
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Journal, issue, pages | Angew. Chem. Int. Ed. Engl., Vol. 60, Page 1220-1226, Year 2021 |
Publish date | Apr 6, 2020 (structure data deposition date) |
Authors | Cui, H. / Divakaran, A. / Pandey, A.K. / Johnson, J.A. / Zahid, H. / Hoell, Z.J. / Ellingson, M.O. / Shi, K. / Aihara, H. / Harki, D.A. / Pomerantz, W.C.K. |
External links | Angew. Chem. Int. Ed. Engl. / PubMed:32975004 |
Methods | X-ray diffraction |
Resolution | 1.53 Å |
Structure data | PDB-6wgx: |
Chemicals | ChemComp-EDO: ChemComp-U0D: ChemComp-HOH: |
Source |
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Keywords | GENE REGULATION/INHIBITOR / BRD4 / GENE REGULATION / GENE REGULATION-INHIBITOR complex |