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-Structure paper
Title | Peptide Inhibitors of Bacterial Protein Synthesis with Broad Spectrum and SbmA-Independent Bactericidal Activity against Clinical Pathogens. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 9590-9602, Year 2020 |
Publish date | Aug 11, 2020 (structure data deposition date) |
![]() | Mardirossian, M. / Sola, R. / Beckert, B. / Valencic, E. / Collis, D.W.P. / Borisek, J. / Armas, F. / Di Stasi, A. / Buchmann, J. / Syroegin, E.A. ...Mardirossian, M. / Sola, R. / Beckert, B. / Valencic, E. / Collis, D.W.P. / Borisek, J. / Armas, F. / Di Stasi, A. / Buchmann, J. / Syroegin, E.A. / Polikanov, Y.S. / Magistrato, A. / Hilpert, K. / Wilson, D.N. / Scocchi, M. |
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Methods | X-ray diffraction |
Resolution | 3 - 3.05 Å |
Structure data | ![]() PDB-7jql: ![]() PDB-7jqm: |
Chemicals | ![]() ChemComp-MG: ![]() ChemComp-ZN: ![]() ChemComp-SF4: ![]() ChemComp-K: ![]() ChemComp-HOH: |
Source |
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![]() | RIBOSOME / Bactenecin 7; antibiotic; 70S ribosome; X-ray structure; inhibition of translation; peptidyl transferase center; nascent peptide exit tunnel |