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-Structure paper
Title | Targeting the trypanosome kinetochore with CLK1 protein kinase inhibitors. |
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Journal, issue, pages | Nat Microbiol, Vol. 5, Page 1207-1216, Year 2020 |
Publish date | Aug 7, 2019 (structure data deposition date) |
Authors | Saldivia, M. / Fang, E. / Ma, X. / Myburgh, E. / Carnielli, J.B.T. / Bower-Lepts, C. / Brown, E. / Ritchie, R. / Lakshminarayana, S.B. / Chen, Y.L. ...Saldivia, M. / Fang, E. / Ma, X. / Myburgh, E. / Carnielli, J.B.T. / Bower-Lepts, C. / Brown, E. / Ritchie, R. / Lakshminarayana, S.B. / Chen, Y.L. / Patra, D. / Ornelas, E. / Koh, H.X.Y. / Williams, S.L. / Supek, F. / Paape, D. / McCulloch, R. / Kaiser, M. / Barrett, M.P. / Jiricek, J. / Diagana, T.T. / Mottram, J.C. / Rao, S.P.S. |
External links | Nat Microbiol / PubMed:32661312 |
Methods | X-ray diffraction |
Resolution | 2.6 Å |
Structure data | PDB-6q2a: |
Chemicals | ChemComp-SO4: ChemComp-5XH: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/TRANSFERASE Inhibitor / kinase / TRANSFERASE-TRANSFERASE Inhibitor complex |