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-Structure paper
Title | Bromodomain-Selective BET Inhibitors Are Potent Antitumor Agents against MYC-Driven Pediatric Cancer. |
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Journal, issue, pages | Cancer Res., Vol. 80, Page 3507-3518, Year 2020 |
Publish date | May 10, 2018 (structure data deposition date) |
![]() | Slavish, P.J. / Chi, L. / Yun, M.K. / Tsurkan, L. / Martinez, N.E. / Jonchere, B. / Chai, S.C. / Connelly, M. / Waddell, M.B. / Das, S. ...Slavish, P.J. / Chi, L. / Yun, M.K. / Tsurkan, L. / Martinez, N.E. / Jonchere, B. / Chai, S.C. / Connelly, M. / Waddell, M.B. / Das, S. / Neale, G. / Li, Z. / Shadrick, W.R. / Olsen, R.R. / Freeman, K.W. / Low, J.A. / Price, J.E. / Young, B.M. / Bharatham, N. / Boyd, V.A. / Yang, J. / Lee, R.E. / Morfouace, M. / Roussel, M.F. / Chen, T. / Savic, D. / Guy, R.K. / White, S.W. / Shelat, A.A. / Potter, P.M. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.05 - 1.5 Å |
Structure data | ![]() PDB-6ddi: ![]() PDB-6ddj: |
Chemicals | ![]() ChemComp-G7V: ![]() ChemComp-SO4: ![]() ChemComp-EDO: ![]() ChemComp-03S: ![]() ChemComp-HOH: |
Source |
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![]() | Transcription/Inhibitor / BET / BRD2 / bromodomain / Inhibitor / Complex / Transcription / Transcription-Inhibitor complex |