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-Structure paper
Title | Discovery of BMS-986251: A Clinically Viable, Potent, and Selective ROR gamma t Inverse Agonist. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 1221-1227, Year 2020 |
Publish date | Feb 5, 2020 (structure data deposition date) |
![]() | Cherney, R.J. / Cornelius, L.A.M. / Srivastava, A. / Weigelt, C.A. / Marcoux, D. / Duan, J.J. / Shi, Q. / Batt, D.G. / Liu, Q. / Yip, S. ...Cherney, R.J. / Cornelius, L.A.M. / Srivastava, A. / Weigelt, C.A. / Marcoux, D. / Duan, J.J. / Shi, Q. / Batt, D.G. / Liu, Q. / Yip, S. / Wu, D.R. / Ruzanov, M. / Sack, J. / Khan, J. / Wang, J. / Yarde, M. / Cvijic, M.E. / Mathur, A. / Li, S. / Shuster, D. / Khandelwal, P. / Borowski, V. / Xie, J. / Obermeier, M. / Fura, A. / Stefanski, K. / Cornelius, G. / Tino, J.A. / Macor, J.E. / Salter-Cid, L. / Denton, R. / Zhao, Q. / Carter, P.H. / Dhar, T.G.M. |
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Methods | X-ray diffraction |
Resolution | 2 Å |
Structure data | ![]() PDB-6vqf: |
Chemicals | ![]() ChemComp-R7V: ![]() ChemComp-GOL: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / RORGT / NUCLEAR HORMONE RECEPTOR / LIGAND-BINDING DOMAIN / INVERSE AGONIST |