+Search query
-Structure paper
Title | Identification of Novel Carbonic Anhydrase IX Inhibitors Using High-Throughput Screening of Pooled Compound Libraries by DNA-Linked Inhibitor Antibody Assay (DIANA). |
---|---|
Journal, issue, pages | SLAS Discov, Vol. 25, Page 1026-1037, Year 2020 |
Publish date | Jun 13, 2019 (structure data deposition date) |
Authors | Tykvart, J. / Navratil, V. / Kugler, M. / Sacha, P. / Schimer, J. / Hlavackova, A. / Tenora, L. / Zemanova, J. / Dejmek, M. / Kral, V. ...Tykvart, J. / Navratil, V. / Kugler, M. / Sacha, P. / Schimer, J. / Hlavackova, A. / Tenora, L. / Zemanova, J. / Dejmek, M. / Kral, V. / Potacek, M. / Majer, P. / Jahn, U. / Brynda, J. / Rezacova, P. / Konvalinka, J. |
External links | SLAS Discov / PubMed:32452709 |
Methods | X-ray diffraction |
Resolution | 1 - 1.38 Å |
Structure data | PDB-6rzx: PDB-6s03: |
Chemicals | ChemComp-ZN: ChemComp-KPQ: ChemComp-HOH: ChemComp-KPW: |
Source |
|
Keywords | LYASE / carbonic anhydrase / inhibitor |