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-Structure paper
Title | Structural and mechanistic insights into 5-lipoxygenase inhibition by natural products. |
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Journal, issue, pages | Nat. Chem. Biol., Vol. 16, Page 783-790, Year 2020 |
Publish date | Nov 14, 2018 (structure data deposition date) |
Authors | Gilbert, N.C. / Gerstmeier, J. / Schexnaydre, E.E. / Borner, F. / Garscha, U. / Neau, D.B. / Werz, O. / Newcomer, M.E. |
External links | Nat. Chem. Biol. / PubMed:32393899 |
Methods | X-ray diffraction |
Resolution | 2.71 - 2.871 Å |
Structure data | PDB-6n2w: PDB-6ncf: |
Chemicals | ChemComp-FE2: ChemComp-30Z: ChemComp-HOH: ChemComp-AF7: |
Source |
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Keywords | OXIDOREDUCTASE/OXIDOREDUCTASE INHIBITOR / Lipoxygenase / inhibitor / allostery / complex / OXIDOREDUCTASE / OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex |