+Search query
-Structure paper
Title | Design and Synthesis of Dihydroxamic Acids as HDAC6/8/10 Inhibitors. |
---|---|
Journal, issue, pages | Chemmedchem, Vol. 15, Page 1163-1174, Year 2020 |
Publish date | Jan 29, 2020 (structure data deposition date) |
![]() | Morgen, M. / Steimbach, R.R. / Geraldy, M. / Hellweg, L. / Sehr, P. / Ridinger, J. / Witt, O. / Oehme, I. / Herbst-Gervasoni, C.J. / Osko, J.D. ...Morgen, M. / Steimbach, R.R. / Geraldy, M. / Hellweg, L. / Sehr, P. / Ridinger, J. / Witt, O. / Oehme, I. / Herbst-Gervasoni, C.J. / Osko, J.D. / Porter, N.J. / Christianson, D.W. / Gunkel, N. / Miller, A.K. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.94301319072 - 2.05 Å |
Structure data | ![]() PDB-6vnq: ![]() PDB-6vnr: |
Chemicals | ![]() ChemComp-R5G: ![]() ChemComp-EDO: ![]() ChemComp-ZN: ![]() ChemComp-K: ![]() ChemComp-PO4: ![]() ChemComp-HOH: |
Source |
|
![]() | Hydrolase/Hydrolase Inhibitor / Histone Deacetylase / Hydrolase-Hydrolase Inhibitor complex / metallohydrolase |