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-Structure paper
Title | Discovery and Optimization of wt-RET/KDR-Selective Inhibitors of RETV804MKinase. |
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Journal, issue, pages | Acs Med. Chem. Lett., Vol. 11, Page 497-505, Year 2020 |
Publish date | Nov 19, 2018 (structure data deposition date) |
Authors | Newton, R. / Waszkowycz, B. / Seewooruthun, C. / Burschowsky, D. / Richards, M. / Hitchin, S. / Begum, H. / Watson, A. / French, E. / Hamilton, N. ...Newton, R. / Waszkowycz, B. / Seewooruthun, C. / Burschowsky, D. / Richards, M. / Hitchin, S. / Begum, H. / Watson, A. / French, E. / Hamilton, N. / Jones, S. / Lin, L.Y. / Waddell, I. / Echalier, A. / Bayliss, R. / Jordan, A.M. / Ogilvie, D. |
External links | Acs Med. Chem. Lett. / PubMed:32292556 |
Methods | X-ray diffraction |
Resolution | 1.88 - 2.05 Å |
Structure data | PDB-6i82: PDB-6i83: |
Chemicals | ChemComp-H6W: ChemComp-EDO: ChemComp-FMT: ChemComp-CL: ChemComp-HOH: ChemComp-H72: |
Source |
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Keywords | ONCOPROTEIN / inhibitor / kinase / proto-oncogene |