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-Structure paper
Title | A New Paroxetine-Based GRK2 Inhibitor Reduces Internalization of themu-Opioid Receptor. |
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Journal, issue, pages | Mol. Pharmacol., Vol. 97, Page 392-401, Year 2020 |
Publish date | Sep 2, 2019 (structure data deposition date) |
![]() | Bouley, R.A. / Weinberg, Z.Y. / Waldschmidt, H.V. / Yen, Y.C. / Larsen, S.D. / Puthenveedu, M.A. / Tesmer, J.J.G. |
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Methods | X-ray diffraction |
Resolution | 2.44 Å |
Structure data | ![]() PDB-6u7c: |
Chemicals | ![]() ChemComp-Q1Y: ![]() ChemComp-MG: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSFERASE/SIGNALING PROTEIN / G-protein coupled receptor kinase / kinase inhibitor / SIGNALING PROTEIN / TRANSFERASE-SIGNALING PROTEIN complex |