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-Structure paper
Title | Garcinoic Acid Is a Natural and Selective Agonist of Pregnane X Receptor. |
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Journal, issue, pages | J. Med. Chem., Vol. 63, Page 3701-3712, Year 2020 |
Publish date | May 21, 2019 (structure data deposition date) |
Authors | Bartolini, D. / De Franco, F. / Torquato, P. / Marinelli, R. / Cerra, B. / Ronchetti, R. / Schon, A. / Fallarino, F. / De Luca, A. / Bellezza, G. ...Bartolini, D. / De Franco, F. / Torquato, P. / Marinelli, R. / Cerra, B. / Ronchetti, R. / Schon, A. / Fallarino, F. / De Luca, A. / Bellezza, G. / Ferri, I. / Sidoni, A. / Walton, W.G. / Pellock, S.J. / Redinbo, M.R. / Mani, S. / Pellicciari, R. / Gioiello, A. / Galli, F. |
External links | J. Med. Chem. / PubMed:32160459 |
Methods | X-ray diffraction |
Resolution | 2.3 Å |
Structure data | PDB-6p2b: |
Chemicals | ChemComp-NQD: ChemComp-DMS: ChemComp-HOH: |
Source |
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Keywords | TRANSCRIPTION / Garcinoic Acid / nuclear receptor |