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-Structure paper
Title | Discovery of Lysine-Targeted eIF4E Inhibitors through Covalent Docking. |
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Journal, issue, pages | J. Am. Chem. Soc., Vol. 142, Page 4960-4964, Year 2020 |
Publish date | Aug 13, 2019 (structure data deposition date) |
![]() | Wan, X. / Yang, T. / Cuesta, A. / Pang, X. / Balius, T.E. / Irwin, J.J. / Shoichet, B.K. / Taunton, J. |
![]() | ![]() ![]() |
Methods | X-ray diffraction |
Resolution | 1.79 - 1.96 Å |
Structure data | ![]() PDB-6u06: ![]() PDB-6u09: |
Chemicals | ![]() ChemComp-EI8: ![]() ChemComp-HOH: ![]() ChemComp-EI9: |
Source |
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![]() | TRANSLATION / cap-binding site / anti-neoplastic / inhibitor / translation initiation blocking / TRANSLATION-INHIBITOR complex / TRANSLATION/INHIBITOR |