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TitleNovel beta- and gamma-Amino Acid-Derived Inhibitors of Prostate-Specific Membrane Antigen.
Journal, issue, pagesJ. Med. Chem., Vol. 63, Page 3261-3273, Year 2020
Publish dateApr 10, 2019 (structure data deposition date)
AuthorsKim, K. / Kwon, H. / Barinka, C. / Motlova, L. / Nam, S. / Choi, D. / Ha, H. / Nam, H. / Son, S.H. / Minn, I. ...Kim, K. / Kwon, H. / Barinka, C. / Motlova, L. / Nam, S. / Choi, D. / Ha, H. / Nam, H. / Son, S.H. / Minn, I. / Pomper, M.G. / Yang, X. / Kutil, Z. / Byun, Y.
External linksJ. Med. Chem. / PubMed:32097010
MethodsX-ray diffraction
Resolution1.76 - 1.77 Å
Structure data

PDB-6rbc:
X-ray structure of human glutamate carboxypeptidase II (GCPII) in complex with a inhibitor KB1157
Method: X-RAY DIFFRACTION / Resolution: 1.77 Å

PDB-6s1x:
X-ray structure of human glutamate carboxypeptidase II (GCPII)-E424M inactive mutant, in complex with a inhibitor KB1160
Method: X-RAY DIFFRACTION / Resolution: 1.76 Å

Chemicals

ChemComp-NAG:
2-acetamido-2-deoxy-beta-D-glucopyranose

ChemComp-ZN:
Unknown entry

ChemComp-CA:
Unknown entry

ChemComp-CL:
Unknown entry

ChemComp-JX5:
(2~{S})-2-[[(2~{R})-2-[4-[(4-iodophenyl)carbonylamino]butanoylamino]-3-oxidanyl-3-oxidanylidene-propyl]carbamoylamino]pentanedioic acid

ChemComp-HOH:
WATER

ChemComp-KRZ:
(2~{S})-2-[[(3~{S})-3-[3-[(4-iodophenyl)carbonylamino]propanoylamino]-4-oxidanyl-4-oxidanylidene-butyl]carbamoylamino]pentanedioic acid

Source
  • homo sapiens (human)
KeywordsHYDROLASE / glutamate carboxypeptidase II (GCPII); NAALADase; prostate-specific membrane antigen; urea-based inhibitor

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