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-Structure paper
Title | Conformation-specific inhibitors of activated Ras GTPases reveal limited Ras dependency of patient-derived cancer organoids. |
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Journal, issue, pages | J. Biol. Chem., Vol. 295, Page 4526-4540, Year 2020 |
Publish date | Jan 28, 2019 (structure data deposition date) |
Authors | Wiechmann, S. / Maisonneuve, P. / Grebbin, B.M. / Hoffmeister, M. / Kaulich, M. / Clevers, H. / Rajalingam, K. / Kurinov, I. / Farin, H.F. / Sicheri, F. / Ernst, A. |
External links | J. Biol. Chem. / PubMed:32086379 |
Methods | X-ray diffraction |
Resolution | 2.9 - 3.15 Å |
Structure data | PDB-6ntc: PDB-6ntd: |
Chemicals | ChemComp-GNP: ChemComp-GOL: ChemComp-MG: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE/PROTEIN BINDING / affinity reagent / RAS inhibitor / TRANSFERASE-PROTEIN BINDING complex / engineered protein |