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-Structure paper
Title | Unexpected CK2 beta-antagonistic functionality of bisubstrate inhibitors targeting protein kinase CK2. |
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Journal, issue, pages | Bioorg. Chem., Vol. 96, Page 103608-103608, Year 2020 |
Publish date | Sep 3, 2019 (structure data deposition date) |
![]() | Pietsch, M. / Viht, K. / Schnitzler, A. / Ekambaram, R. / Steinkruger, M. / Enkvist, E. / Nienberg, C. / Nickelsen, A. / Lauwers, M. / Jose, J. ...Pietsch, M. / Viht, K. / Schnitzler, A. / Ekambaram, R. / Steinkruger, M. / Enkvist, E. / Nienberg, C. / Nickelsen, A. / Lauwers, M. / Jose, J. / Uri, A. / Niefind, K. |
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Methods | X-ray diffraction |
Resolution | 1.599 - 1.994 Å |
Structure data | ![]() PDB-6spw: ![]() PDB-6spx: |
Chemicals | ![]() ChemComp-NA: ![]() ChemComp-A0Z: ![]() ChemComp-HOH: ![]() ChemComp-9AB: |
Source |
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![]() | TRANSFERASE / protein kinase CK2 casein kinase 2 bisubstrate inhibitor |