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TitleElucidation of an Allosteric Mode of Action for a Thienopyrazole ROR gamma t Inverse Agonist.
Journal, issue, pagesChemmedchem, Vol. 15, Page 561-565, Year 2020
Publish dateDec 3, 2019 (structure data deposition date)
Authorsde Vries, R.M.J.M. / Doveston, R.G. / Meijer, F.A. / Brunsveld, L.
External linksChemmedchem / PubMed:32053744
MethodsX-ray diffraction
Resolution2.321 Å
Structure data

PDB-6tlm:
ROR(gamma)t ligand binding domain in complex with allosteric ligand compound 13 (Glenmark)
Method: X-RAY DIFFRACTION / Resolution: 2.321 Å

Chemicals

ChemComp-MJE:
4-[1-[2,6-bis(chloranyl)phenyl]carbonyl-5-methyl-thieno[3,2-c]pyrazol-3-yl]benzoic acid

ChemComp-HOH:
WATER

Source
  • homo sapiens (human)
KeywordsGENE REGULATION / Nuclear Receptor / Allosteric / Inverse Agonist / Inhibitor

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