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-Structure paper
Title | Structure-guided design of pure orthosteric inhibitors of alpha IIb beta 3 that prevent thrombosis but preserve hemostasis. |
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Journal, issue, pages | Nat Commun, Vol. 11, Page 398-398, Year 2020 |
Publish date | Dec 5, 2018 (structure data deposition date) |
Authors | Adair, B.D. / Alonso, J.L. / van Agthoven, J. / Hayes, V. / Ahn, H.S. / Yu, I.S. / Lin, S.W. / Xiong, J.P. / Poncz, M. / Arnaout, M.A. |
External links | Nat Commun / PubMed:31964886 |
Methods | X-ray diffraction |
Resolution | 3.1 Å |
Structure data | PDB-6naj: |
Chemicals | ChemComp-NAG: ChemComp-MN: ChemComp-HOH: |
Source |
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Keywords | CELL ADHESION / HYBRID DOMAIN / PSI / EGF REPEATS / BETA TAIL / CALF / THIGH / BETA PROPELLER / RGD MOTIF / FIBRONECTIN / VITRONECTIN |