+Search query
-Structure paper
Title | Evaluating the Advantages of Using 3D-Enriched Fragments for Targeting BET Bromodomains. |
---|---|
Journal, issue, pages | Acs Med. Chem. Lett., Vol. 10, Page 1648-1654, Year 2019 |
Publish date | Nov 2, 2019 (structure data deposition date) |
Authors | Johnson, J.A. / Nicolaou, C.A. / Kirberger, S.E. / Pandey, A.K. / Hu, H. / Pomerantz, W.C.K. |
External links | Acs Med. Chem. Lett. / PubMed:31857841 |
Methods | X-ray diffraction |
Resolution | 1.307 - 1.51 Å |
Structure data | PDB-6uvj: PDB-6uvm: PDB-6uwx: |
Chemicals | ChemComp-EDO: ChemComp-DMS: ChemComp-QJ1: ChemComp-HOH: ChemComp-QJA: ChemComp-QKD: |
Source |
|
Keywords | GENE REGULATION/INHIBITOR / BRD4(D1) / inhibitor / GENE REGULATION-INHIBITOR complex |